Endoxifen (E-isomer)
CAS No. 114828-90-9
Endoxifen (E-isomer) ( E-Endoxifen; Endoxifen E-isomer )
Catalog No. M26199 CAS No. 114828-90-9
Endoxifen E-isomer is the E-isomer of (Z)-Endoxifen. Endoxifen E-isomer has antiestrogenic effects.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 155 | Get Quote |
|
10MG | 230 | Get Quote |
|
25MG | 462 | Get Quote |
|
50MG | 740 | Get Quote |
|
100MG | 1161 | Get Quote |
|
200MG | Get Quote | Get Quote |
|
500MG | Get Quote | Get Quote |
|
1G | Get Quote | Get Quote |
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Biological Information
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Product NameEndoxifen (E-isomer)
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NoteResearch use only, not for human use.
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Brief DescriptionEndoxifen E-isomer is the E-isomer of (Z)-Endoxifen. Endoxifen E-isomer has antiestrogenic effects.
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DescriptionEndoxifen E-isomer is the E-isomer of (Z)-Endoxifen. Endoxifen E-isomer has antiestrogenic effects.(In Vitro):Endoxifen exists as the potently anti-estrogenic (Z)-isomer and the lesser-known (E)-isomer. (E)-Endoxifen is identified as the primary degradant. The (E)-isomer is an impurity in (Z)-Endoxifen drug substance and increases under certain storage conditions.
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SynonymsE-Endoxifen; Endoxifen E-isomer
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PathwayEndocrinology/Hormones
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TargetEstrogen Receptor/ERR
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RecptorPEGs
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Research Area——
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Indication——
Chemical Information
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CAS Number114828-90-9
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Formula Weight373.5
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Molecular FormulaC25H27NO2
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Purity>98% (HPLC)
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Solubility——
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SMILESOC1=CC=C(/C(C2=CC=C(OCCNC)C=C2)=C(C3=CC=CC=C3)/CC)C=C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.An S, et al. Small-molecule PROTACs:An emerging and promising approach for the development of targeted therapy drugs. EBioMedicine. 2018 Oct;36:553-562.
molnova catalog
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